Recent advances in transition metal-catalyzed Csp2-monofluoro-, difluoro-, perfluoromethylation and trifluoromethylthiolation
G. Landelle, A. Panossian, S. Pazenok, J.-P. Vors, F. R. Leroux
Beilstein J. Org. Chem. 2013, 9, 2476-2536.
Want create site? Find Free WordPress Themes and plugins.
Before 2014
Manfred Schlosser (1934-2013)
F. Leroux
Angew. Chem. Int. Ed. 2013, 52, 12483.
Convenient and Reliable Routes Towards 2-Aminothiazoles: Palladium-catalyzed versus Copper-catalyzed Aminations of Halothiazoles
S. Toulot, T. Heinrich, F. R. Leroux
Adv. Synth. Catal. 2013, 355, 3263-3272.
Atropodiastereoselective C-H Olefination of Biphenyl p-Tolylsulfoxides with Acrylates
T. Wesch, F. R. Leroux, F. Colobert
Adv. Synth. Cat. 2013, 355, 2139-2144.
Synthesis and structural properties of an hexaaza[5]helicene containing two [1,2,3]triazolo[1,5-a]pyridine moieties
R. Adam, R. Ballesteros-Garrido, O. Vallcorba, B. Abarca, R. Ballesteros, F. R. Leroux, F. Colobert, J. M. Amigó, J. Rius
Tetrahedron Lett. 2013, 54, 4316-4319.
A New Life for an Old Reagent: Fluoroalkyl Amino Reagents as Efficient Tools for the Synthesis of Diversely Fluorinated Pyrazoles
S. Pazenok, F. Giornal, G. Landelle, N. Lui, J.-P. Vors, F. R. Leroux
Eur. J. Org. Chem. 2013, 4249-4253.
Palladium-Catalyzed Intramolecular Direct Arylation of 2-Bromo-diaryl Sulfoxides via C–H Bond Activation
T. Wesch, A. Berthelot-Bréhier, F. R. Leroux, F. Colobert
Org. Lett. 2013, 15, 2490-2493.
Synthesis of diversely fluorinated pyrazoles as novel active agrochemical ingredients
F. Giornal, S. Pazenok, L. Rodefeld, N. Lui, J.-P. Vors, F. R. Leroux
J. Fluorine Chem. 2013, 152, 2-11.
Transition Metal-Free Atropo-selective Synthesis of Biaryl Compounds Based on Arynes
F. R. Leroux, A. Berthelot, L. Bonnafoux, A. Panossian, F. Colobert
Chem. Eur. J. 2012, 18, 14232-14236.
Stereoselective Synthesis of P-Chirogenic Dibenzophosphole (boranes) via Aryne Intermediates
V. Diemer, A. Berthelot, J. Bayardon, S. Jugé, F. R. Leroux, F. Colobert
J. Org. Chem. 2012, 77, 6117–6127.
Stereoselective Synthesis of o-Bromo (or Iodo)aryl P-Chirogenic Phosphines owing to the Aryne Chemistry
J. Bayardon, H. Laureano, V. Diemer,M. Dutartre, U. Das, Y. Rousselin, J.-C. Henry, F. Colobert, F. R. Leroux, S. Jugé
J. Org. Chem. 2012, 77, 5759-5769.
Triazolopyridines. Part 28. The ring–chain isomerization strategy: triazolopyridine- and triazoloquinoline–pyridine based fluorescence ligands
R. Ballesteros-Garrido, E. Delgado-Pinar, B. Abarca, R. Ballesteros, F. R. Leroux, F. Colobert, R. J. Zaragoza, E. Garcia-Espana
Tetrahedron 2012, 68, 3701-3707.
Construction of the biaryl-part of vancomycin aglycon via atropo- 10Q1 diastereoselective Suzuki–Miyaura coupling
T. Leermann, P.-E. Broutin, F. R. Leroux, F. Colobert
Org. Biomol. Chem. 2012, 10, 4095-4102.
Aryne-mediated Fluorination : Synthesis of Fluorinated Biaryls via a Sequential Desilylation – Halide Elimination – Fluoride Addition Process
V. Diemer, J. S. Garcia, F. R. Leroux, F. Colobert
J. Fluorine Chem. 2012, 134, 146-155.
Polar Organometallic Chemistry
F. R. Leroux
Catalytic Palladium-Phosphination: Modular Synthesis of C1-Symmetric Biaryl-Based Diphosphines
L. Bonnafoux, R. Gramage-Doria, F. Colobert, F. R. Leroux
Chem. Eur. J. 2011, 11008-11016.
Bromine-Lithium Exchange : An Efficient Tool in the Modular Construction of Biaryl Ligands
L. Bonnafoux, F. R. Leroux, F. Colobert
Beilstein J. Org. Chem. 2011, 7, 1278-1287.
Highly Efficient One-pot Access to Functionalized Arylboronic Acids via Non-cryogenic Bromine/Magnesium Exchanges
T. Leermann, F. R. Leroux, F. Colobert
Org. Lett. 2011, 13, 4479-4481.
Through-Space J(P,P) and J(P,F) Spin Spin Coupling in C1-Symmetric Biaryl Diphosphines
L. Bonnafoux, L. Ernst, F. R. Leroux, F. Colobert
Eur. J. Inorg. Chem. 2011, 3387-3397.
Efficient and Complementary Methods Offering Access to Synthetically Valuable 1,2-Dibromobenzenes
V. Diemer, F. R. Leroux, F. Colobert
Eur. J. Org. Chem. 2011, 327-340.
Regioselectivity in the ARYNE Cross Coupling of Aryllithiums with Functionalized 1,2-Dibromobenzenes
V. Diemer, M. Begaud, F. R. Leroux, F. Colobert
Eur. J. Org. Chem. 2011, 341-354.
[1,2,3]Triazolo[1,5-a]pyridyl Phosphines Reflecting the Influence of Phosphorus Lone Pair Orientation on Spectroscopic Properties
R. Ballesteros-Garrido, L. Bonnafoux, F. Blanco, R. Ballesteros, F. R. Leroux, B. Abarca, F. Colobert, I. Alkorta, J. Elguero
Dalton Trans. 2011, 40, 1387-1395.
2,2′,6-Tribromobiphenyl via the Transition-metal Free ARYNE Coupling: A Valuable Tool in the Synthesis of Biphenyls
L. Bonnafoux, F. Colobert, F. R. Leroux
Synlett 2010, 2953-2955.
A General and Recommendable Approach Towards Trifluoromethoxy Pyridines: First X-ray Structure Determinations and Quantum Chemistry Studies
B. Manteau, P. Genix, S. Pazenok, J.-P. Vors, F. Giornal, C. Leuenberger, F. R. Leroux
Eur. J. Org. Chem. 2010, 6043-6066.
Efficient Synthesis of Quaternary and P-Stereogenic Phosphonium Triflates
E. Rémond, A. Tessier, F. R. Leroux, J. Bayardon, S. Jugé
Org. Lett. 2010, 12, 1568-1571.
New Trends in the Chemistry of a-Fluorinated Ethers, Thioethers, Amines and Phosphines
B. Manteau, S. Pazenok, J.-P. Vors, F. R. Leroux
J. Fluorine Chem. 2010, 131, 140-158.
Axial Chirality Control During Suzuki-Miyaura Cross-coupling Reactions: The t-Butylsulfinyl Group as an Efficient Chiral Auxiliary
F. Colobert, V. Valdivia, S. Choppin, F. R. Leroux, I. Fernández, E. Álvarez,N. Khiar
Org. Lett. 2009, 11, 5130-5133.
Publications Selected by Synfacts 2010
3-(2-Pyridyl)-[1,2,3]Triazolo[1,5-a]quinoline. A Theoretical and Experimental Analysis of Ring-Chain Isomerisation
R. Ballesteros-Garrido, F. Blanco, R. Ballesteros, F. R. Leroux, B. Abarca, F. Colobert, I. Alkorta, J. Elguero
Eur. J. Org. Chem. 2009, 5765-5778.
[1,2,3]Triazolo[1,5-a]pyridine Derivatives as Molecular Chemosensors for Zinc(II), Nitrite and Cyanide
R. Ballesteros-Garrido, B. Abarca, R. Ballesteros, F. R. Leroux, F. Colobert, E. Garcia-Espana
New J. Chem. 2009, 2102-2106.
The [1,2,3]Triazolo[1,5-a]pyridine Ring: A Sensitive Sensor for the Electronic Profile of Phosphor(III) Substituents
R. Ballesteros-Garrido, L. Bonnafoux, F. R. Leroux, B. Abarca, F. Colobert
Dalton Trans. 2009, 5068-5070.
The Deprotonative Metalation of [1,2,3]Triazolo[1,5-a]uinolone. Synthesis of 8-Haloquinolin-2-Carboxaldehydes
R. Ballesteros-Garrido, F. R. Leroux, R. Ballesteros, B. Abarca, F. Colobert
Tetrahedron 2009, 65, 4410-4417.
Triazolopyridines. Part 26. The preparation of novel [1,2,3]triazolo[1,5-a]pyridine sulfoxides
B. Abarca, R. Ballesteros, R. Ballesteros-Garrido, F. Colobert, F. R. Leroux
Tetrahedron 2008, 64, 3794-3801.
Trifluoromethyl Ethers – Synthesis and Properties of an Unusual Substituent
F. R. Leroux, B. Manteau, J.-P. Vors, S. Pazenok
Beilstein J. Org. Chem. 2008, 4, 13.
Relative Carbanion Basicity as Driving Force for an Intramolecular Silyl Migration of Lithiated Biphenyls
L. Bonnafoux, R. Scopelliti, F. R. Leroux, F. Colobert
Tetrahedron Lett. 2007, 48, 8768-8772.
A Practical Transition-metal-free Aryl-Aryl Coupling Method : Arynes as Key Intermediates
F. R. Leroux, L. Bonnafoux, C. Heiss, F. Colobert, D. A. Lanfranchi
Adv. Synth. Catal. 2007, 349, 2705-2713.
Triazolopyridines. Part 25. Synthesis of new chiral ligands from [1,2,3]triazolo[1,5-a]pyridines
B. Abarca, R. Ballesteros, R. Ballesteros-Garrido, F. Colobert, F. R. Leroux
Tetrahedron 2007, 63, 10479-10485.
Efficient First Palladium-Catalyzed Synthesis of Heteroaromatic Sulfoxides
F. Colobert, R. Ballesteros-Garrido, F. R. Leroux, R. Ballesteros, B. Abarca
Tetrahedron Lett. 2007, 48, 6896-6899.
a-Fluorinated Ethers as “Exotic” Entity in Medicinal Chemistry
P. Jeschke, E. Baston, F. R. Leroux
Mini-Rev. Med. Chem. 2007, 7, 1027-1034.
The First Stereoselective Pd-catalyzed Addition of Boronic Acids onto Aldehydes
A. Novodomská, M. Dudiková, F. R. Leroux, F. Colobert
Tetrahedron: Asymmetry 2007, 18, 1628-1634.
Publications Selected by Synfacts 2007
First Modular Synthesis of Dissymetric Biaryldiphosphine Ligands Allowing Tunable Steric and Electronic Effects
F. R. Leroux, H. Mettler
Adv. Synth. Cat. 2007, 349, 323-336.
Inhibitors of Steroidal Cytochrome P450 Enzymes as Targets for Drug Development
E. Baston, F. R. Leroux
Recent Pat. Anti-Cancer Drug Discovery 2007, 2, 31-58.
A Highly Efficient Low Temperature Modification of the Classical Ullmann Reaction
F. R. Leroux, R. Simon, N. Nicod
Lett. Org. Chem. 2006, 3, 948-954.
Fluorine Modulated Biaryls : How Does the Smallest Heteroelement Affect Atropisomerism
F. Leroux
Chimica Oggi/Chemistry Today 2006, 24, 9-11.
New Vistas in Halogen/Metal Exchange Reactions : The Discrimination between Seemingly Equal Halogens
F. Leroux, N. Nicod, L. Bonnafoux, B. Quissac, F. Colobert
Lett. Org. Chem. 2006, 3, 165-169.
Ligand Tailoring : The First Modular Synthesis of Atropisomeric Biarylligands
F. Leroux, H. Mettler
Synlett 2006, 766-770.
The Effect of Ring Size on Reactivity : The Diagnostic Value of “Rate Profiles”
E. Masson, F. Leroux
Helv. Chim. Acta 2005, 88, 1375-1386.
Inhibition of P450 17 as a New Strategie for the Treatment of Prostate Cancer
F. Leroux
Curr. Med. Chem. 2005, 12, 1623-1629.
α-Fluorinated Ethers, Thioethers and Amines : Anomerically Biased Species
F. Leroux, P. Jeschke, M. Schlosser
Chem. Rev. 2005, 105, 827-856.
Palladium-Catalyzed Borylation of Phenyl Bromides and Application in One-Pot Suzuki-Miyaura Biphenyl Synthesis
P.-E. Broutin, I. Čerňa, M. Campaniello, F. Leroux, F. Colobert
Org. Lett. 2004, 6, 4419-4422.
Atropisomerism, Biphenyls and Fluorine : A Comparison of Torsional Barriers and Twist Angles
F. Leroux
ChemBioChem 2004, 5, 644-649.
The Remarkable Configurational Stability of ortho, ortho’-Tetrafluoro Substituted Biphenyls : 2,2’,4,4’,6,6’-Hexafluorobiphenyl-3,3’-dicarboxylic Acid as a Model
F. Leroux, M. Maurin, N. Nicod, R. Scopelliti
Tetrahedron Lett. 2004, 45, 1899-1902.
N-(4-Biphenylmethyl)imidazoles as Potential Therapeutics for the Treatment of Prostate Cancer : Metabolic Robustness Due to Fluorine Substitution ?
F. Leroux, T. Hutschenreuter, C. Charrière, R. Scopelliti, R.W. Hartmann
Helv. Chim. Acta 2003, 86, 2671-2686.
Did you find apk for android? You can find new Free Android Games and apps.